OX1 receptor 选择性拮抗剂

目录号	产品详情
S1545	SB408124 SB408124 is a non-peptide antagonist for OX1 receptor with K_i of 57 nM and 27 nM in both whole cell and membrane, respectively, exhibits 50-fold selectivity over OX2 receptor.
S7585	SB-334867 SB-334867 is a selective orexin-1 (OX1) receptor antagonist.
S2160	Almorexant HCl Almorexant HCl (ACT-078573) is an orally active, dual orexin receptor antagonist with IC50 of 6.6 nM and 3.4 nM for OX1 and OX2 receptor, respectively. Phase 3.

目录号

产品详情

S1545

SB408124 is a non-peptide antagonist for OX1 receptor with K_i of 57 nM and 27 nM in both whole cell and membrane, respectively, exhibits 50-fold selectivity over OX2 receptor.

S7585

SB-334867

SB-334867 is a selective orexin-1 (OX1) receptor antagonist.

S2160

Almorexant HCl

Almorexant HCl (ACT-078573) is an orally active, dual orexin receptor antagonist with IC50 of 6.6 nM and 3.4 nM for OX1 and OX2 receptor, respectively. Phase 3.